SCHEMBL18640508

SCHEMBL18640508

C[C@@H]1c2ccc(Br)cc2CN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMK2A Q9UQM7 1/20 0.42
KIF11 P52732 1/20 0.40
HSD17B3 P37058 3/20 0.40
SRD5A1 P18405 2/20 0.36
AKR1C3 P42330 2/20 0.36
SRD5A2 P31213 1/20 0.36
BRD4 O60885 1/20 0.36
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
ADRA2A P08913 1/20 0.34
PNMT P11086 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
DRD1 P21728 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16099073 1.00 CAMK2A (0.42) CAMK2AKIF11HSD17B3SRD5A1AKR1C3
SCHEMBL28764376 0.85 CAMK2A (0.46) CAMK2ASRD5A1AKR1C3DRD1
SCHEMBL2898555 0.84 KIF11 (0.38) CAMK2AKIF11HSD17B3SRD5A1BRD4
SCHEMBL2917359 0.84 KIF11 (0.38) CAMK2AKIF11HSD17B3SRD5A1BRD4
SCHEMBL18940029 0.83 CAMK2A (0.46) CAMK2AKIF11HSD17B3SRD5A1AKR1C3
SCHEMBL2121418 0.82 CAMK2A (0.40) CAMK2AKIF11HSD17B3SRD5A1AKR1C3
SCHEMBL18940076 0.81 KIF11 (0.40) CAMK2AKIF11HSD17B3SRD5A1AKR1C3
SCHEMBL28386200 0.80 NR1H2 (0.42) ABHD6
SCHEMBL29410655 0.80 NR1H2 (0.42) ABHD6
SCHEMBL16099540 0.80 NR1H2 (0.42) ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017046605-A1 ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2017-03-23 WO disclosed
WO-2017046606-A1 ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2017-03-23 WO disclosed