SCHEMBL18652013

SCHEMBL18652013

OCC(COCc1ccccc1)COc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.47
CA2 P00918 2/20 0.47
CA7 P43166 2/20 0.47
CA9 Q16790 2/20 0.47
TSHR P16473 1/20 0.45
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HIF1A Q16665 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TACR1 P25103 2/20 0.42
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
LTA4H P09960 1/20 0.41
EPHX2 P34913 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14453897 0.89 CA1 (0.56) CA1CA2CA7CA9TSHR
SCHEMBL14453900 0.86 CA1 (0.53) CA1CA2CA7CA9TSHR
SCHEMBL1865158 0.86 CA1 (0.56) CA1CA2CA7CA9TSHR
SCHEMBL24304919 0.82 LMNA (0.57) LMNAPTGS1
SCHEMBL23483165 0.80 GSTP1 (0.46) CA1CA2CA7CA9TSHR
SCHEMBL6068726 0.79 CA1 (0.50) CA1CA2CA7CA9TSHR
SCHEMBL9662754 0.79 CA1 (0.64) CA1CA2CA7CA9TSHR
SCHEMBL10052085 0.79 CA1 (0.50) CA1CA2CA7CA9TSHR
SCHEMBL6068730 0.79 CA1 (0.50) CA1CA2CA7CA9TSHR
SCHEMBL300081 0.79 CA1 (0.64) CA1CA2CA7CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632457-B1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2017-03-22 EP disclosed