SCHEMBL18654078

SCHEMBL18654078

C=CC[C@@H](C(=O)N1C(=O)OC[C@@H]1c1ccccc1)[C@H](C)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
IL6ST P40189 1/20 0.39
IDH1 O75874 9/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RIPK1 Q13546 1/20 0.37
NAAA Q02083 1/20 0.36
CYP2C19 P33261 1/20 0.36
AVPR1A P37288 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796721 0.85 ALDH1A1 (0.44) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL16796724 0.85 ALDH1A1 (0.44) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930233 0.84 ALDH1A1 (0.39) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930237 0.84 ALDH1A1 (0.39) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930236 0.84 ALDH1A1 (0.39) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930584 0.84 IL6ST (0.45) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930588 0.84 IL6ST (0.45) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930586 0.84 IL6ST (0.45) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930715 0.83 ALDH1A1 (0.39) ALDH1A1GAAHTTIL6STIDH1
SCHEMBL21930717 0.83 ALDH1A1 (0.39) ALDH1A1GAAHTTIL6STIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595483-B1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2017-03-22 EP disclosed