SCHEMBL18657449

SCHEMBL18657449

COc1cc(N2CCNCC2)c(N)cc1Nc1ncc(Cl)c(OC2CN(S(C)(=O)=O)C2)n1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 9/20 0.48
EGFR P00533 8/20 0.46
LRRK2 Q5S007 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196875 0.91 EGFR (0.51) ALKEGFRLRRK2
SCHEMBL18657447 0.85 EGFR (0.55) ALKEGFR
SCHEMBL17196873 0.79 EGFR (0.55) ALKEGFRLRRK2
SCHEMBL17196683 0.77 EGFR (0.65) ALKEGFR
SCHEMBL18563173 0.75 EGFR (0.55) ALKEGFR
SCHEMBL17196871 0.75 EGFR (0.46) ALKEGFRLRRK2
SCHEMBL17196684 0.75 EGFR (0.66) EGFR
SCHEMBL18563178 0.73 EGFR (0.61) EGFR
Formic Acid SCHEMBL18549295 0.73 EGFR (0.64) EGFR
SCHEMBL17196834 0.71 EGFR (0.66) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3144292-B1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (US) 2020-08-26 EP disclosed
EP-3144292-A1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD (US) 2017-03-22 EP disclosed