SCHEMBL18670976

SCHEMBL18670976

CC(C)c1ccc(C(=O)Nc2cc(-c3ccccc3)cnc2N)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.56
LDHB P07195 1/20 0.56
GSK3B P49841 1/20 0.55
HDAC1 Q13547 10/20 0.51
HDAC2 Q92769 8/20 0.49
HDAC3 O15379 7/20 0.49
NCOR2 Q9Y618 6/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
MAP4K4 O95819 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18670987 0.85 HDAC1 (0.54) LDHALDHBGSK3BHDAC1HDAC2
SCHEMBL18670955 0.83 GSK3B (0.55) LDHALDHBGSK3BHDAC1HDAC2
SCHEMBL2227269 0.81 CHEK2 (0.62) GSK3BHDAC1HDAC2HDAC3MAP4K4
SCHEMBL18653509 0.81 HDAC2 (0.75) HDAC1HDAC2HDAC3
SCHEMBL18670971 0.81 GSK3B (0.53) GSK3BHDAC1HDAC2HDAC3
SCHEMBL20806967 0.81 CA1 (0.44) LDHALDHBGSK3BHDAC1TP53
SCHEMBL27810689 0.81 HDAC1 (0.53) GSK3BHDAC1HDAC2HDAC3
SCHEMBL18670958 0.81 HDAC1 (0.71) GSK3BHDAC1HDAC2HDAC3NCOR2
SCHEMBL3646469 0.79 HDAC1 (0.60) GSK3BHDAC1HDAC2HDAC3
SCHEMBL3777895 0.77 HDAC1 (0.54) GSK3BHDAC1HDAC2HDAC3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9603950-B1 Compounds of imaging agent with HDAC inhibitor for treatment of Alzheimer syndrome and method of synthesis thereof INSTITUTE OF NUCLEAR ENERGY RESEARCH (TW) 2017-03-28 US disclosed
US-9603950-B1 Compounds of imaging agent with HDAC inhibitor for treatment of Alzheimer syndrome and method of synthesis thereof INSTITUTE OF NUCLEAR ENERGY RESEARCH (TW) 2017-03-28 US disclosed