SCHEMBL1868066

SCHEMBL1868066

CCCn1c(Oc2cc(C)ccn2)nc(=O)c2c1N=C(C1CCCC1)[N]2

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 15/20 0.38
ADORA2B P29275 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA3 P0DMS8 1/20 0.35
CRHR1 P34998 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1864786 0.87 ADORA1 (0.39) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1869240 0.83 ADORA1 (0.38) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1871420 0.83 ADORA1 (0.41) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1868690 0.82 ADORA1 (0.57) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1875306 0.81 ADORA1 (0.56) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1875998 0.81 ADORA1 (0.38) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1864689 0.81 ADORA1 (0.44) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1866236 0.80 ADORA1 (0.41) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1861450 0.80 ADORA1 (0.49) ADORA1ADORA2BADORA2AADORA3
SCHEMBL1874917 0.80 ADORA1 (0.57) ADORA1ADORA2BADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP disclosed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO disclosed