SCHEMBL18686087

SCHEMBL18686087

CCCc1nn(C)c2c(=O)nc(-c3cc(N(C)C4CCN(C(=O)OC(C)(C)C)CC4)ccc3OCC)[nH]c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.56
HDAC1 Q13547 14/20 0.56
HDAC6 Q9UBN7 14/20 0.56
HDAC2 Q92769 6/20 0.56
HDAC3 O15379 1/20 0.56
NCOR2 Q9Y618 1/20 0.56
PDE6C P51160 3/20 0.44
PDE3A Q14432 3/20 0.43
PDE3B Q13370 2/20 0.43
PDE2A O00408 1/20 0.41
ABCC4 O15439 1/20 0.41
ABCC5 O15440 1/20 0.41
PDE6D O43924 1/20 0.41
PDE8A O60658 1/20 0.41
PDE9A O76083 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
PDE6A P16499 1/20 0.41
PDE6G P18545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17390117 0.89 PDE5A (0.70) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL31174348 0.77 PDE5A (0.55) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL17390216 0.75 PDE5A (0.68) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL17390124 0.74 PDE5A (0.75) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL22558019 0.74 KMT2A (0.62) PDE5APDE6CPDE3APDE3BPDE2A
SCHEMBL22793623 0.73 KMT2A (0.60) PDE5APDE6CPDE3APDE3BPDE2A
SCHEMBL17390135 0.72 PDE5A (0.64) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL17017276 0.72 PDE5A (0.54) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL17404873 0.72 PDE5A (1.00) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL18069562 0.71 PDE5A (0.65) PDE5AHDAC1HDAC6HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2961741-B1 NOVEL COMPOUNDS AS DUAL INHIBITORS OF PHOSPHODIESTERASES AND HISTONE DEACETYLASES FUND PARA LA INVESTIG MEDICA APLICADA (ES) 2017-04-05 EP disclosed