SCHEMBL18697646

SCHEMBL18697646

Cc1noc(-c2cc(F)ccc2C(=O)N2CCC[C@@H](Nc3ccc(C(F)(F)F)cn3)C2)n1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.72
HCRTR2 O43614 5/20 0.66
MAP3K12 Q12852 2/20 0.46
OPRK1 P41145 1/20 0.44
JAK2 O60674 1/20 0.44
JAK3 P52333 1/20 0.44
GFER P55789 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144777 1.00 HCRTR1 (0.72) HCRTR1HCRTR2MAP3K12OPRK1JAK2
SCHEMBL20145089 0.92 HCRTR1 (0.62) HCRTR1HCRTR2MAP3K12OPRK1JAK2
SCHEMBL20144963 0.92 HCRTR1 (0.62) HCRTR1HCRTR2MAP3K12OPRK1JAK2
SCHEMBL20144856 0.90 HCRTR1 (0.66) HCRTR1HCRTR2MAP3K12OPRK1JAK2
SCHEMBL20144938 0.90 HCRTR1 (0.66) HCRTR1HCRTR2MAP3K12OPRK1JAK2
SCHEMBL20144772 0.85 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL17506064 0.84 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL16031159 0.84 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL20144885 0.83 HCRTR1 (0.69) HCRTR1HCRTR2
SCHEMBL17510802 0.79 HCRTR1 (1.00) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed
US-9611251-B2 Substituted piperidine compounds and their use as orexin receptor modulators JANSSEN PHARMACEUTICA NV (BE) 2017-04-04 US disclosed