SCHEMBL20144856

SCHEMBL20144856

Cc1noc(-c2ccccc2C(=O)N2CCCC(Nc3ccc(C(F)(F)F)cn3)C2)n1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.66
HCRTR2 O43614 7/20 0.52
MAP3K12 Q12852 1/20 0.49
JAK2 O60674 1/20 0.45
JAK3 P52333 1/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
OPRK1 P41145 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144938 1.00 HCRTR1 (0.66) HCRTR1HCRTR2MAP3K12JAK2JAK3
SCHEMBL18697646 0.90 HCRTR1 (0.72) HCRTR1HCRTR2MAP3K12JAK2JAK3
SCHEMBL20144777 0.90 HCRTR1 (0.72) HCRTR1HCRTR2MAP3K12JAK2JAK3
SCHEMBL1835677 0.83 KDM4E (0.52) HCRTR1HCRTR2MAP3K12LMNA
SCHEMBL16030811 0.83 HCRTR1 (0.82) HCRTR1HCRTR2
SCHEMBL1141302 0.82 MAP3K12 (0.51) HCRTR1HCRTR2MAP3K12
SCHEMBL1141304 0.82 MAP3K12 (0.51) HCRTR1HCRTR2MAP3K12
SCHEMBL20145089 0.81 HCRTR1 (0.62) HCRTR1HCRTR2MAP3K12JAK2JAK3
SCHEMBL20144963 0.81 HCRTR1 (0.62) HCRTR1HCRTR2MAP3K12JAK2JAK3
SCHEMBL17028118 0.80 HCRTR1 (1.00) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed