SCHEMBL1869909

SCHEMBL1869909

CC[C@@]1(CNC(C)=O)OC2(C=C(C(=O)O)C(S(=O)(=O)Nc3ccc(F)cc3Cl)CC2)O[C@H]1CNC(C)=O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 5/20 0.44
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
KMT2A Q03164 1/20 0.32
CNR2 P34972 1/20 0.31
MRGPRX1 Q96LB2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15093794 0.86 TLR4 (0.47) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL1866347 0.86 TLR4 (0.47) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL1862851 0.86 TLR4 (0.47) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL4159467 0.85 TLR4 (0.48) TLR4PSEN1PSEN2APH1BNCSTN
SCHEMBL1862994 0.83 TLR4 (0.47) TLR4KMT2AMRGPRX1
SCHEMBL1863031 0.83 TLR4 (0.46) TLR4NPC1RAB9AKMT2AMRGPRX1
SCHEMBL1864588 0.83 TLR4 (0.46) TLR4NPC1RAB9AKMT2AMRGPRX1
SCHEMBL1862043 0.81 TLR4 (0.48) TLR4KMT2AMRGPRX1
SCHEMBL1864173 0.80 TLR4 (0.43) TLR4MRGPRX1
SCHEMBL1864310 0.79 TLR4 (0.61) TLR4LMNAKMT2AMRGPRX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7935835-B2 Substituted cycloalkene derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-05-03 US disclosed