SCHEMBL1870650

SCHEMBL1870650

CC(C)(C)[S@+]([O-])NCCCCc1ccc(Br)nc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.33
NFKB1 P19838 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP11B1 P15538 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1134880 0.96 NFKB1 (0.34) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL22886675 0.81 CYP11B1 (0.35) CYP11B1
SCHEMBL31639522 0.81 CYP11B1 (0.35) CYP11B1
SCHEMBL17441145 0.80 AR (0.33)
SCHEMBL17441143 0.80 AR (0.33)
SCHEMBL1419592 0.76 AR (0.34)
SCHEMBL1870915 0.76 AR (0.34)
SCHEMBL21591858 0.76 ESR1 (0.46)
SCHEMBL21591855 0.74 PREP (0.34)
SCHEMBL17441501 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed
WO-2011056440-A1 HETEROCYCLIC COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-05-12 WO disclosed