SCHEMBL18726258

SCHEMBL18726258

NC(=O)c1cc(-c2ccc(Br)cc2)n[nH]1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACR P10323 2/20 0.57
SNCA P37840 1/20 0.56
ALPL P05186 9/20 0.55
RAB9A P51151 2/20 0.53
NPC1 O15118 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CA12 O43570 4/20 0.53
TP53 P04637 1/20 0.51
RPA1 P27694 1/20 0.51
MAPT P10636 4/20 0.51
PLA2G10 O15496 1/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
CA9 Q16790 2/20 0.48
POLB P06746 1/20 0.48
CASP1 P29466 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23803931 0.85 ALPL (0.73) ACRSNCAALPLRAB9ANPC1
SCHEMBL2846632 0.83 ALPL (0.73) ACRALPLCA12TP53RPA1
SCHEMBL4638840 0.83 ALPL (0.73) ACRALPLCA12TP53RPA1
SCHEMBL29444415 0.83 ALPL (0.73) ACRSNCAALPLRAB9ACA12
SCHEMBL2789578 0.83 TP53 (0.74) ACRALPLCA12TP53RPA1
SCHEMBL2851298 0.83 SCN9A (0.54) ACRALPLRAB9ANPC1SMN1; SMN2
SCHEMBL4789868 0.81 CCNC (0.54) ALPLCA12TP53RPA1MAPT
SCHEMBL855912 0.80 ALPL (0.76) SNCAALPLRAB9ANPC1SMN1; SMN2
SCHEMBL20661049 0.80 TP53 (0.51) ACRALPLRAB9ACA12TP53
SCHEMBL2848443 0.80 ALPL (0.76) ACRALPLRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114057646-B Pyrazole derivative and application thereof in preparation of antitumor drugs 常州大学 2023-05-02 CN disclosed
CN-114057646-A Pyrazole derivative and application thereof in preparation of antitumor drugs 常州大学 2022-02-18 CN disclosed
EP-2376478-B1 PYRIDYLOXYINDOLES INHIBITORS OF VEGF-R2 AND USE THEREOF FOR TREATMENT OF DISEASE NOVARTIS AG (CH) 2017-04-19 EP disclosed