SCHEMBL18746102

SCHEMBL18746102

BC(=O)Nc1c(C)noc1-c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 5/20 0.49
LPAR3 Q9UBY5 3/20 0.49
MAPT P10636 4/20 0.47
KDM4E B2RXH2 1/20 0.47
ABCC3 O15438 1/20 0.42
ABCC4 O15439 1/20 0.42
ABCB11 O95342 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2C9 P11712 1/20 0.42
ABCB4 P21439 1/20 0.42
ABCC2 Q92887 1/20 0.42
SLCO1B3 Q9NPD5 1/20 0.42
SLCO1B1 Q9Y6L6 1/20 0.42
SMPD1 P17405 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LPAR2 Q9HBW0 2/20 0.41
ALDH1A1 P00352 2/20 0.40
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6003 0.88 LPAR1 (0.54) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL2761525 0.84 LPAR1 (0.57) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL11389 0.81 NPC1 (0.51) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL2761399 0.81 LPAR1 (0.54) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL1345 0.80 LPAR1 (0.53) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL2761476 0.80 LPAR1 (0.65) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL6434 0.79 LPAR1 (0.49) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL18597709 0.79 LPAR1 (0.40) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL2761269 0.78 LPAR1 (0.63) LPAR1LPAR3MAPTKDM4EABCC3
SCHEMBL12973654 0.78 LPAR1 (0.63) LPAR1LPAR3MAPTKDM4EABCC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9624182-B2 Compounds as lysophosphatidic acid receptor antagonists AMIRA PHARMACEUTICALS, INC. (US) 2017-04-18 US disclosed