SCHEMBL2761525

SCHEMBL2761525

COC(=O)Nc1c(C)noc1-c1ccc(Br)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 5/20 0.57
LPAR3 Q9UBY5 3/20 0.57
ABCC3 O15438 1/20 0.48
ABCC4 O15439 1/20 0.48
ABCB11 O95342 1/20 0.48
CYP2C8 P10632 1/20 0.48
CYP2C9 P11712 1/20 0.48
ABCB4 P21439 1/20 0.48
ABCC2 Q92887 1/20 0.48
SLCO1B3 Q9NPD5 1/20 0.48
SLCO1B1 Q9Y6L6 1/20 0.48
LPAR2 Q9HBW0 2/20 0.47
MAPT P10636 3/20 0.46
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.45
RAB9A P51151 2/20 0.42
TNIK Q9UKE5 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761399 0.88 LPAR1 (0.54) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL6003 0.87 LPAR1 (0.54) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL2761476 0.87 LPAR1 (0.65) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL1345 0.87 LPAR1 (0.53) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL2761269 0.85 LPAR1 (0.63) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL12973654 0.85 LPAR1 (0.63) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL18746102 0.84 LPAR1 (0.49) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL12973580 0.83 LPAR1 (0.60) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL15897508 0.83 LPAR1 (0.60) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL2761499 0.83 LPAR1 (0.49) LPAR1LPAR3ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010141768-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed
WO-2010141768-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed