SCHEMBL18746342

SCHEMBL18746342

COC(O)c1cc(C(F)(F)F)ccc1Nc1ccc2c(ccn2Cc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.48
KCNQ2 O43526 2/20 0.48
KCNQ4 P56696 2/20 0.48
KCNQ5 Q9NR82 2/20 0.48
ERBB2 P04626 5/20 0.45
EGFR P00533 3/20 0.42
ERBB4 Q15303 1/20 0.42
NR1I2 O75469 1/20 0.41
CDK1 P06493 1/20 0.40
CDK4 P11802 1/20 0.40
CCNB1 P14635 1/20 0.40
CCND1 P24385 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CDK6 Q00534 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
P2RX7 Q99572 1/20 0.39
EPHX2 P34913 1/20 0.38
PPARD Q03181 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15712533 0.83 KCNQ3 (0.53) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL15712529 0.80 KCNQ3 (0.54) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL17067712 0.75 EGFR (0.41) ERBB2EGFRERBB4NR1I2HDAC3
SCHEMBL15712561 0.71 ERBB2 (0.51) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL17067776 0.71 SYK (0.49) ERBB2EGFRERBB4CDK1CDK4
SCHEMBL17067816 0.71 EGFR (0.43) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL15712122 0.71 ERBB2 (0.48) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL20850689 0.71 ERBB2 (0.48) KCNQ3KCNQ2KCNQ4KCNQ5ERBB2
SCHEMBL15712210 0.71 ERBB2 (0.48) ERBB2EGFRERBB4NR1I2CDK1
SCHEMBL15712256 0.70 ERBB2 (0.46) ERBB2EGFRERBB4NR1I2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9624215-B2 Amine derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2017-04-18 US disclosed