SCHEMBL18751636

SCHEMBL18751636

Cc1ccc(C(=O)NC2(c3ccc4cnccc4n3)CC2)cc1-c1ccc2oc(-c3ccc(F)cc3)c(C=O)c2c1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.59
CYP3A4 P08684 5/20 0.59
KCNH2 Q12809 3/20 0.57
NR1I2 O75469 1/20 0.57
MAPK14 Q16539 3/20 0.39
LCK P06239 1/20 0.39
CSF1R P07333 1/20 0.39
KDR P35968 1/20 0.39
ABL1 P00519 7/20 0.37
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12330955 0.94 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL143691 0.89 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL12330701 0.86 CYP2C8 (0.62) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL145125 0.83 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL141259 0.82 CYP2C8 (0.72) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL2471972 0.80 CYP2C8 (0.58) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL143480 0.78 CYP2C8 (0.77) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2471970 0.77 CYP2C8 (0.54) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL18752118 0.76 CYP2C8 (0.56) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL120717 0.76 CYP2C8 (0.79) CYP2C8CYP3A4KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-04-19 EP disclosed