SCHEMBL2471972

SCHEMBL2471972

CNC(=O)c1c(-c2cc(C(=O)NC3(c4ccc5cnccc5n4)CC3)ccc2C)ccc2oc(-c3ccc(F)cc3)cc12

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.58
CYP3A4 P08684 5/20 0.58
KCNH2 Q12809 3/20 0.56
NR1I2 O75469 1/20 0.56
MAPK14 Q16539 2/20 0.36
LCK P06239 1/20 0.36
CSF1R P07333 1/20 0.36
KDR P35968 1/20 0.36
IDO1 P14902 2/20 0.33
ABL1 P00519 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL143691 0.88 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL2471646 0.88 CYP2C8 (0.62) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL141259 0.87 CYP2C8 (0.72) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL2471970 0.85 CYP2C8 (0.54) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL145125 0.83 CYP2C8 (0.75) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL143635 0.81 CYP2C8 (0.72) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL18751636 0.80 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL120472 0.78 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL142368 0.78 CYP2C8 (0.78) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL143480 0.77 CYP2C8 (0.77) CYP2C8CYP3A4KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112769-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed