SCHEMBL18752129

SCHEMBL18752129

Cc1c(F)cc(C(=O)NC2(c3nc4cnccc4o3)CC2)cc1-c1ccc2oc(-c3ccc(F)cc3)c(C=O)c2c1F

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.47
KCNH2 Q12809 3/20 0.47
CYP3A4 P08684 5/20 0.43
NR1I2 O75469 1/20 0.38
ABL1 P00519 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31
MAPK13 O15264 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
APEX1 P27695 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
IDO1 P14902 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL119435 0.89 CYP2C8 (0.61) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL120775 0.82 CYP2C8 (0.63) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL19401445 0.81 CYP2C8 (0.55) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL12330957 0.81 CYP2C8 (0.51) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL19401368 0.80 CYP2C8 (0.55) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL119462 0.79 CYP2C8 (0.74) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL119399 0.78 CYP2C8 (0.59) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL143315 0.77 CYP2C8 (0.60) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL120472 0.76 CYP2C8 (0.59) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL120828 0.74 CYP2C8 (0.77) CYP2C8KCNH2CYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545051-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-04-19 EP disclosed