SCHEMBL19401445

SCHEMBL19401445

Cc1c(F)cc(C(=O)NC2(c3ncccn3)CC(F)(F)C2)cc1-c1ccc2oc(-c3ccc(F)cc3)c(C=O)c2c1F

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.55
KCNH2 Q12809 3/20 0.55
CYP3A4 P08684 5/20 0.47
NR1I2 O75469 1/20 0.41
ABL1 P00519 1/20 0.33
ACKR3 P25106 1/20 0.31
IDO1 P14902 2/20 0.31
CYP2C9 P11712 4/20 0.31
MAPK14 Q16539 4/20 0.31
MAPK11 Q15759 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19401368 0.91 CYP2C8 (0.55) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL19401316 0.90 CYP2C8 (0.68) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL19385895 0.88 CYP2C8 (0.71) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL12330957 0.84 CYP2C8 (0.51) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL2143062 0.81 CYP2C8 (0.82) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL19401443 0.81 CYP2C8 (0.67) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL19401314 0.81 CYP2C8 (0.69) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL18752129 0.81 CYP2C8 (0.47) CYP2C8KCNH2CYP3A4NR1I2ABL1
SCHEMBL15285746 0.80 CYP2C8 (0.72) CYP2C8KCNH2CYP3A4NR1I2
SCHEMBL9899509 0.80 CYP2C8 (0.72) CYP2C8KCNH2CYP3A4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017165233-A1 BENZOFURAN DERIVATIVES FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-28 WO disclosed