SCHEMBL18754397

SCHEMBL18754397

Cc1nc2cccc(C)n2c1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.58
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 4/20 0.46
POLB P06746 2/20 0.46
CYP1A2 P05177 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
TP53 P04637 7/20 0.40
PKM P14618 6/20 0.40
PKLR P30613 5/20 0.40
GAA P10253 10/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
MAPT P10636 6/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
PPP1CA P62136 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPK1 P28482 1/20 0.35
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8374902 0.81 HTT (0.43) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL11157649 0.79 HTT (0.42) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL16506289 0.79 HTT (0.54) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL16506921 0.79 HTT (0.43) HTTALDH1A1KDM4EPOLBCYP1A2
Bromide SCHEMBL10919771 0.78 HTT (0.49) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL11356063 0.76 HTT (0.70) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL21863678 0.76 HTT (0.51) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL21849002 0.76 HTT (0.51) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL21894539 0.75 KDM4E (0.55) HTTALDH1A1KDM4EPOLBCYP1A2
SCHEMBL22275503 0.75 HTT (0.50) HTTALDH1A1KDM4EPOLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017214269-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2017-12-14 WO disclosed
EP-3036235-B1 NEW BIS-AMIDO PYRIDINES BOEHRINGER INGELHEIM INT (DE) 2017-04-19 EP disclosed