SCHEMBL18754654

SCHEMBL18754654

COC(=O)C1C[C@H](Oc2ccc(F)cc2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.52
HRH3 Q9Y5N1 3/20 0.51
KCNH2 Q12809 1/20 0.51
MCL1 Q07820 12/20 0.45
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
PTPN1 P18031 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29523156 1.00 P2RX3 (0.52) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL12442648 1.00 P2RX3 (0.52) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL18617461 1.00 P2RX3 (0.52) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL6846802 0.90 P2RX3 (0.53) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL6846804 0.90 P2RX3 (0.53) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL25365111 0.90 P2RX3 (0.53) P2RX3MCL1NR1H2NR1H3
SCHEMBL23632505 0.89 P2RX3 (0.51) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL23632277 0.89 P2RX3 (0.51) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL23632438 0.89 P2RX3 (0.51) P2RX3HRH3KCNH2MCL1NR1H2
SCHEMBL23632270 0.89 P2RX3 (0.51) P2RX3HRH3KCNH2MCL1NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534170-B1 IAP BIR DOMAIN BINDING COMPOUNDS PHARMASCIENCE INC (CA) 2017-04-19 EP disclosed