SCHEMBL1875599

SCHEMBL1875599

C[C@H](OC(=O)C(O)(c1cccs1)c1cccs1)C1CCCN1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 15/20 0.43
CHRM2 P08172 13/20 0.43
CHRM1 P11229 11/20 0.43
CHRM4 P08173 2/20 0.40
CHRM5 P08912 1/20 0.40
TSPO P30536 1/20 0.40
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
OPRK1 P41145 1/20 0.40
KCNH2 Q12809 1/20 0.40
PDE3A Q14432 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SLC6A3 Q01959 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
DHFR P00374 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1880296 0.82 CHRM3 (0.46) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL1873958 0.81 SLC6A3 (0.44) CHRM3CHRM2KCNH2SLC6A3SLC6A2
SCHEMBL1878142 0.81 SLC6A3 (0.44) CHRM3CHRM2KCNH2SLC6A3SLC6A2
SCHEMBL9671210 0.71 SLC6A3 (0.36) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL20476343 0.69 CHRM3 (0.55) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL27861451 0.69 SLC6A3 (0.40) SLC6A3SLC6A2SLC6A4DHFR
SCHEMBL2596407 0.68 CHRM3 (0.57) CHRM3CHRM2CHRM1CHRM4CHRM5
Acetic Acid SCHEMBL20476349 0.68 CHRM3 (0.54) CHRM3CHRM2CHRM1CHRM4CHRM5
SCHEMBL826276 0.68 CHRM3 (0.49) CHRM3CHRM2CHRM1CHRM4CHRM5
Fluoride SCHEMBL14940626 0.67 CHRM3 (0.56) CHRM3CHRM2CHRM1CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947730-B2 Piperidinium and pyrrolidinium derivatives as ligands for the muscarinic M3 receptor NOVARTIS AG (CH) 2011-05-24 US disclosed