SCHEMBL18756376

SCHEMBL18756376

Cc1nc(C(=O)NC2CCCC2)cc(Cc2ccc(Cl)nc2)c1C

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 8/20 0.47
CYP3A4 P08684 1/20 0.43
CYP3A5 P20815 1/20 0.43
CNR1 P21554 4/20 0.43
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18756664 0.99 CHRM1 (0.46) CHRM1CYP3A4CYP3A5CNR1
SCHEMBL18756570 0.89 CHRM1 (0.46) CHRM1CYP3A4CYP3A5CNR1
SCHEMBL18725353 0.88 CHRM1 (0.61) CHRM1CNR1
SCHEMBL18756663 0.88 CHRM1 (0.61) CHRM1CNR1
SCHEMBL18725457 0.86 CHRM1 (0.61) CHRM1
SCHEMBL6893880 0.85 CHRM1 (0.54) CHRM1
SCHEMBL12073429 0.84 PARP1 (0.44) CHRM1CNR1
SCHEMBL2224496 0.84 GAA (0.55) CHRM1CNR1
SCHEMBL18756200 0.83 CNR1 (0.46) CHRM1CYP3A4CNR1
SCHEMBL22212629 0.82 CHRM1 (0.48) CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3156397-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2017-04-19 EP disclosed