SCHEMBL18758786

SCHEMBL18758786

O=C(O)CNc1ccc2c([N+](=O)[O-])cccc2c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MAPT P10636 5/20 0.45
POLB P06746 2/20 0.44
APEX1 P27695 1/20 0.44
CASP6 P55212 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PLCG2 P16885 2/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7487865 0.85 TDP1 (0.51) ALDH1A1MAPTPOLBCASP6NPC1
SCHEMBL18740461 0.82 ALDH1A1 (0.40) ALDH1A1MAPTPOLBNPC1RAB9A
SCHEMBL8973925 0.81 KMT2A (0.49) ALDH1A1APEX1MAPK1TDP1
SCHEMBL8168105 0.76 EGFR (0.59) ALDH1A1MAPTPOLBSMN1; SMN2L3MBTL1
SCHEMBL3948505 0.75 MAPT (0.51) ALDH1A1MAPTAPEX1L3MBTL1TDP1
SCHEMBL6192945 0.74 MAPT (0.61) ALDH1A1MAPTPOLBSMN1; SMN2L3MBTL1
SCHEMBL1797099 0.74 MAPT (0.61) ALDH1A1MAPTPOLBSMN1; SMN2L3MBTL1
SCHEMBL11052022 0.74 PTPN1 (0.58) ALDH1A1POLBAPEX1CASP6TDP1
SCHEMBL20839720 0.73 KMT2A (0.67) ALDH1A1MAPTRAB9ASMN1; SMN2L3MBTL1
SCHEMBL809030 0.73 ALDH1A1 (0.60) ALDH1A1MAPTPOLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017063755-A1 CONFORMATIONALLY CONSTRAINED MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2017-04-20 WO disclosed
WO-2017063754-A1 CONFORMATIONALLY CONSTRAINED MACROCYCLIC COMPOUNDS AS PIN1 MODULATORS POLYPHOR AG (CH) 2017-04-20 WO disclosed