SCHEMBL18780403

SCHEMBL18780403

COc1cc(CCN[C@H](C)C=O)c(Cl)cc1NC(=O)Nc1cnc(C#N)cn1

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 20/20 0.76
AURKA O14965 1/20 0.65
CDK2 P24941 1/20 0.65
FLT4 P35916 1/20 0.65
FLT3 P36888 1/20 0.65
MAPKAPK2 P49137 1/20 0.65
GSK3A P49840 1/20 0.65
GSK3B P49841 1/20 0.65
RPS6KA3 P51812 1/20 0.65
MAPK12 P53778 1/20 0.65
CDK5 Q00535 1/20 0.65
STK3 Q13188 1/20 0.65
ROCK1 Q13464 1/20 0.65
CAMK1 Q14012 1/20 0.65
MAPKAPK3 Q16644 1/20 0.65
PRKD2 Q9BZL6 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18780302 1.00 CHEK1 (0.76) CHEK1AURKACDK2FLT4FLT3
SCHEMBL18780355 0.87 CHEK1 (0.76) CHEK1AURKACDK2FLT4FLT3
SCHEMBL2593415 0.86 CHEK1 (1.00) CHEK1
SCHEMBL16206653 0.84 CHEK1 (0.88) CHEK1FLT4FLT3RPS6KA3PRKD2
SCHEMBL16206635 0.84 CHEK1 (0.88) CHEK1FLT4FLT3RPS6KA3PRKD2
SCHEMBL14965385 0.84 CHEK1 (0.74) CHEK1AURKACDK2FLT4FLT3
Hydrochloric Acid SCHEMBL17684931 0.84 CHEK1 (0.86) CHEK1FLT4FLT3RPS6KA3PRKD2
SCHEMBL2589904 0.84 CHEK1 (1.00) CHEK1
Hydrochloric Acid SCHEMBL17684925 0.84 CHEK1 (0.86) CHEK1FLT4FLT3RPS6KA3PRKD2
Hydrochloric Acid SCHEMBL16195313 0.83 CHEK1 (0.73) CHEK1AURKACDK2FLT4FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9630931-B2 Pharmaceutically active pyrazine derivatives SENTINEL ONCOLOGY LIMITED (GB) 2017-04-25 US disclosed