SCHEMBL1880644

SCHEMBL1880644

COc1c(O)ccc2cc[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA12 O43570 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
BRD4 O60885 3/20 0.37
TNF P01375 1/20 0.36
RIPK1 Q13546 1/20 0.36
PPARG P37231 1/20 0.35
APP P05067 1/20 0.35
MAPT P10636 1/20 0.35
BCHE P06276 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9315235 0.80 BCHE (0.35) ESR1MEN1KMT2ABRD4TNF
SCHEMBL30261030 0.78 BRD4 (0.45) MEN1POLBMAPK1KMT2ABRD4
SCHEMBL7835424 0.78 BRD4 (0.45) MEN1POLBMAPK1KMT2ABRD4
SCHEMBL20354829 0.77 AHR (0.47) MEN1POLBMAPK1KMT2ABRD4
SCHEMBL2305754 0.77 BRD4 (0.41) MEN1POLBMAPK1KMT2ABRD4
SCHEMBL1162240 0.75 KDM4E (0.42) CA1CA12CA7CA9POLB
SCHEMBL28878115 0.75 KEAP1 (0.53) MEN1POLBMAPK1KMT2AMAPT
SCHEMBL15550121 0.74 KEAP1 (0.40) MEN1POLBMAPK1KMT2ABRD4
SCHEMBL8055277 0.74 TNF (0.39) ESR1ESR2BRD4TNFRIPK1
SCHEMBL9315426 0.73 MCL1 (0.42) MEN1POLBMAPK1KMT2ABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 150 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103517703-B Stain and application thereof 天野酶制品株式会社 2016-11-09 CN claimed
EP-2623093-B1 DYE FOR KERATIN FIBERS USING BILIRUBIN OXIDASE AND INDOLE DERIVATIVES AMANO ENZYME INC (JP) 2016-05-25 EP claimed
CN-103998016-B Employ the dyeing of the keratin fiber of indole analog AMANO ENZYME INC. (JP) 2015-09-16 CN claimed
CN-103408554-B Hypertensive activity reducing pyrrole coumarins compound and preparation method thereof UNIV XI AN JIAOTONG 2015-07-08 CN claimed
US-20140359950-A1 DYEING OF KERATIN FIBERS USING INDOLE ANALOGUE AMANO ENZYME INC. (JP) 2014-12-11 US claimed
CN-103408554-A Hypertensive activity reducing pyrrole coumarins compound and preparation method thereof UNIV XI AN JIAOTONG 2013-11-27 CN claimed
EP-0597022-B2 PROCESS FOR THE TEMPORARY DYEING OF KERATIN FIBRES INVOLVING AN INSOLUBLE PIGMENT OBTAINED BY THE OXIDATIVE POLYMERISATION OF INDOLE DERIVATIVES OREAL (FR) 1999-11-17 EP claimed
US-5874091-A PROTECTION OF SKIN AND HAIR AGAINST ULTRAVIOLET RADIATION AND FOR PIGMENTATION OF THE SKIN AND HAIR; HOMOGENEOUS AQUEOUS DISPERSION OF LAMELLAR AND ENCAPSULATING VESICLES; STORAGE STABILITY; STORING MELANIN PIGMENT IN THE STRATUM CORNEUM. L'OREAL (FR) 1999-02-23 US claimed
EP-0587837-B1 Cosmetic composition containing melanistic pigments in association with certain tocopherols, and method for protecting the skin, the hair, the mucous membranes and cosmetic compositions OREAL (FR) 1998-06-03 EP claimed
EP-0544874-B1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS OREAL (FR) 1998-04-08 EP claimed
WO-1993000068-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-01-07 WO claimed
EP-0518773-A1 Cosmetic composition containing a blend of metallic oxids nanopigments and melanic pigments L'OREAL (FR) 1992-12-16 EP claimed
EP-0504347-A1 COSMETIC COMPOSITION COMPRISING A DISPERSION OF LIPIDIC VESICLES AS WELL AS MELANIC PIGMENTS. OREAL (FR) 1992-09-23 EP claimed
EP-0500446-A1 Skin-tanning composition containing indole derivatives and dihydroxyacetone L'OREAL (FR) 1992-08-26 EP claimed
WO-1992005761-A1 COSMETIC COMPOSITION COMPRISING A DISPERSION OF LIPIDIC VESICLES AS WELL AS MELANIC PIGMENTS L'OREAL (FR) 1992-04-16 WO claimed
EP-0467767-A1 Product based on flaky particles containing melanine pigment and process for their preparation L'OREAL (FR) 1992-01-22 EP claimed
EP-0446132-A1 Keratinous fibres dyeing process with 6 or 7-monohydroxyindols at acidic pH and compositions L'OREAL (FR) 1991-09-11 EP claimed
EP-0428442-A1 Composition comprising derivatives of 6- or 7-hydroxyindole as couplers and dyeing processes using same L'OREAL (FR) 1991-05-22 EP claimed
EP-0379409-A1 Products based on polymer particles containing melanine pigments, process for their preparation, and their use, particularly cosmetically L'OREAL (FR) 1990-07-25 EP claimed
EP-0376776-A2 Process for dyeing keratinous fibres with hydroxyindole associated with quinone and 1,4-benzoquinone L'OREAL (FR) 1990-07-04 EP claimed