SCHEMBL18809491

SCHEMBL18809491

O=C(NC12CC(C1)C2)c1ccccc1F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
MAPT P10636 2/20 0.60
HPGD P15428 2/20 0.60
KDM4E B2RXH2 1/20 0.60
TSHR P16473 1/20 0.60
ALOX12 P18054 1/20 0.60
HTT P42858 1/20 0.60
ATM Q13315 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HSD17B10 Q99714 1/20 0.60
CNR2 P34972 8/20 0.55
FAAH O00519 4/20 0.55
GAA P10253 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CNR1 P21554 2/20 0.49
NPC1 O15118 1/20 0.49
HSD11B1 P28845 1/20 0.47
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26240417 0.88 KDM4E (0.58) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL31419639 0.80 GAA (0.51) ALDH1A1MAPTHPGDHTTGAA
SCHEMBL30848463 0.80 HPGD (0.60) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL24268174 0.79 KDM4E (0.59) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL26240424 0.77 GRM5 (0.52) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL30848467 0.76 CNR2 (0.89) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL31191005 0.75 TSHR (1.00) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL15121240 0.75 TSHR (1.00) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL10928771 0.75 KDM4E (0.72) ALDH1A1MAPTHPGDKDM4ETSHR
SCHEMBL3709144 0.74 KDM4E (0.70) ALDH1A1MAPTHPGDKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970174-B1 FUSED FURANS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2017-05-03 EP disclosed