SCHEMBL18822011

SCHEMBL18822011

COC(=O)Nc1ccc2c(c1)NC(=O)CCCCC(C(=O)O)c1nc-2c(C)[nH]1

nearest known ligand 0.62

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
F11 P03951 20/20 0.62
KLK1 P06870 14/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18822013 0.90 F11 (0.59) F11KLK1
SCHEMBL22294599 0.89 F11 (0.62) F11KLK1
SCHEMBL23049437 0.89 F11 (0.62) F11KLK1
SCHEMBL24220218 0.88 F11 (0.62) F11KLK1
SCHEMBL24220096 0.83 F11 (0.53) F11KLK1
SCHEMBL18822005 0.82 F11 (0.51) F11KLK1
SCHEMBL18822542 0.81 F11 (0.56) F11KLK1
SCHEMBL18822365 0.80 F11 (0.51) F11KLK1
SCHEMBL18822360 0.80 F11 (0.65) F11KLK1
SCHEMBL614075 0.79 F11 (0.56) F11KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017074833-A1 MACROCYCLIC SPIROCARBAMATE DERIVATIVES AS FACTOR XIA INHIBITORS, PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2017-05-04 WO disclosed