SCHEMBL1882298

SCHEMBL1882298

Cc1cccc2cc(CCl)c(-c3ccccc3)nc12

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
PIK3CD O00329 13/20 0.47
ATM Q13315 1/20 0.46
PDE10A Q9Y233 1/20 0.41
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1598508 0.85 PIK3CD (0.53) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL1887862 0.85 MEN1 (0.48) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL1884319 0.85 PIK3CD (0.47) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL3386976 0.82 PIK3CD (0.46) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL1597713 0.81 PIK3CD (0.65) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL28539195 0.80 PDE10A (0.62) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL1598030 0.80 PIK3CD (0.49) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL3654574 0.80 PIK3CD (0.44) L3MBTL1DRD4DRD3PIK3CDATM
SCHEMBL1878444 0.79 PIK3CD (0.51) L3MBTL1DRD4DRD3PIK3CDATM
Formic Acid SCHEMBL1887914 0.78 PIK3CD (0.45) L3MBTL1DRD4DRD3PIK3CDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231641-B1 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-06-01 EP disclosed
US-8399483-B2 Quinoxaline and quinoline derivatives as kinase inhibitors UCB PHARMA S.A. (BE) 2013-03-19 US disclosed
US-20110105508-A1 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA, S.A. (BE) 2011-05-05 US disclosed
EP-2231641-A2 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS UCB Pharma, S.A. (BE) 2010-09-29 EP disclosed
WO-2009081105-A2 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105508-A1 QUINOXALINE AND QUINOLINE DERIVATIVES AS KINASE INHIBITORS PDXK, PDPK1, PIKFYVE L3MBTL1 3240/4885DRD4 3720/4885DRD3 2440/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.