SCHEMBL18828640

SCHEMBL18828640

CCOC(=O)[C@H]1CC1c1ccc(C(F)(F)F)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.52
KCNH2 Q12809 1/20 0.44
SSTR4 P31391 3/20 0.41
HDAC4 P56524 1/20 0.39
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNQ4 P56696 1/20 0.39
KCNQ5 Q9NR82 1/20 0.39
SSTR1 P30872 1/20 0.37
LIPE Q05469 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
LTC4S Q16873 1/20 0.36
DGAT1 O75907 1/20 0.36
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15797825 1.00 HRH3 (0.52) HRH3KCNH2SSTR4HDAC4KCNQ3
SCHEMBL15797826 1.00 HRH3 (0.52) HRH3KCNH2SSTR4HDAC4KCNQ3
SCHEMBL15805108 1.00 HRH3 (0.52) HRH3KCNH2SSTR4HDAC4KCNQ3
SCHEMBL15805085 1.00 HRH3 (0.52) HRH3KCNH2SSTR4HDAC4KCNQ3
SCHEMBL1473448 0.89 HRH3 (0.40) HRH3MAPTPKM
SCHEMBL15314513 0.86 HRH3 (0.55) HRH3KCNH2SSTR4HDAC4SSTR1
SCHEMBL451266 0.86 HRH3 (0.55) HRH3KCNH2SSTR4HDAC4SSTR1
SCHEMBL455274 0.86 HRH3 (0.55) HRH3KCNH2SSTR4HDAC4SSTR1
SCHEMBL12128172 0.86 HRH3 (0.55) HRH3KCNH2SSTR4HDAC4SSTR1
SCHEMBL15797832 0.83 KDM1A (0.44) MAPTPKMKDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2931708-B1 CYCLOPROPYLBORONIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF DIVERCHIM (FR) 2017-05-10 EP disclosed