SCHEMBL18834880

SCHEMBL18834880

Cn1c(=O)n(CCCO)c(=O)c2[nH]c(Cl)nc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.46
ADORA2B P29275 3/20 0.46
PDE4A P27815 2/20 0.46
PDE4B Q07343 2/20 0.46
PDE4C Q08493 2/20 0.46
PDE4D Q08499 2/20 0.46
ADORA1 P30542 3/20 0.45
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
KMT2A Q03164 1/20 0.43
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
ADRA2A P08913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16029024 0.86 ADORA2B (0.50) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL3114983 0.85 ADORA1 (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL18834910 0.84 PDE2A (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL16027743 0.83 ADORA2A (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL3121598 0.83 ADORA1 (0.53) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL3121149 0.81 ADORA1 (0.52) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL29430494 0.81 ADORA2B (0.49) ADORA2AADORA2BALDH1A1LMNACYP1A2
SCHEMBL3120638 0.80 ADORA2B (0.49) ADORA2AADORA2BPDE4APDE4BPDE4C
SCHEMBL3112561 0.80 ADORA2B (0.64) ADORA2AADORA2BADORA1ADORA3ALDH1A1
SCHEMBL21499663 0.79 ADORA2A (0.48) ADORA2AADORA2BPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970303-B1 SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF HYDRA BIOSCIENCES INC (US) 2017-05-10 EP disclosed