SCHEMBL18845331

SCHEMBL18845331

CCCN(CCc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
TP53 P04637 1/20 0.42
AOC3 Q16853 1/20 0.42
PRSS1 P07477 1/20 0.42
CTSG P08311 1/20 0.42
CTRB1 P17538 1/20 0.42
CMA1 P23946 1/20 0.42
CTSK P43235 3/20 0.42
SIGMAR1 Q99720 1/20 0.42
DRD2 P14416 1/20 0.41
OPRM1 P35372 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25047708 0.92 HDAC3 (0.48) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL4781274 0.90 HDAC3 (0.48) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL4450404 0.89 BCHE (0.55) HDAC3HDAC1HDAC2NCOR2L3MBTL1
SCHEMBL1845666 0.88 MEN1 (0.46) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL2260891 0.87 MEN1 (0.45) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL9060170 0.87 HDAC1 (0.60) HDAC3HDAC1HDAC2NCOR2L3MBTL1
SCHEMBL9823156 0.87 HDAC1 (0.54) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL25046666 0.86 L3MBTL1 (0.45) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL3050230 0.85 MEN1 (0.46) HDAC3HDAC1HDAC2NCOR2MEN1
SCHEMBL25047881 0.85 L3MBTL1 (0.47) HDAC3HDAC1HDAC2NCOR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017079476-A1 LSD1 INHIBITORS Mirati Therapeutics, Inc. (US) 2017-05-11 WO disclosed