SCHEMBL1884680

SCHEMBL1884680

CC(C)c1cc(C(=O)O)c(Cc2ccccc2)n1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.51
FABP4 P15090 1/20 0.46
CCR2 P41597 1/20 0.41
TSHR P16473 2/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HNF4A P41235 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HTT P42858 1/20 0.39
PTPN1 P18031 2/20 0.39
PTPN2 P17706 1/20 0.39
PTPN6 P29350 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GPR35 Q9HC97 1/20 0.39
IDH1 O75874 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1887819 0.89 NOTUM (0.51) NOTUMFABP4CCR2TSHRLMNA
SCHEMBL1880517 0.87 MAPT (0.47) NOTUMTSHRSMN1; SMN2ALDH1A1KDM4E
SCHEMBL1884573 0.84 NOTUM (0.47) NOTUM
SCHEMBL12672207 0.83 NOTUM (0.49) NOTUMFABP4CCR2TSHRLMNA
SCHEMBL1875610 0.83 NOTUM (0.46) NOTUMFABP4CCR2TSHRLMNA
SCHEMBL1873898 0.82 NOTUM (0.54) NOTUMFABP4CCR2TSHRLMNA
SCHEMBL1875953 0.82 NOTUM (0.70) NOTUMFABP4CCR2TSHRLMNA
SCHEMBL1880515 0.79 S1PR3 (0.63)
SCHEMBL3756783 0.77 NOTUM (0.44) NOTUMCCR2TSHRLMNASMN1; SMN2
SCHEMBL1880697 0.76 NOTUM (0.50) NOTUMFABP4CCR2TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110105567-A1 Pyrrole Compounds Having Sphingosine-1-Phosphate Receptor Agonist Or Antagonist Biological Activity ALLERGAN, INC. (US) 2011-05-05 US disclosed
EP-2185506-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2010-05-19 EP disclosed
WO-2009026407-A1 PYRROLE COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST OR ANTAGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2009-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105567-A1 Pyrrole Compounds Having Sphingosine-1-Phosphate Receptor Agonist Or Antagonist Biological Activity S1PR1, S1PR2, S1PR3 NOTUM 822/4885FABP4 952/4885CCR2 396/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.