SCHEMBL1884692

SCHEMBL1884692

COc1ccc(NC(N)=S)cc1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.53
MAPT P10636 4/20 0.53
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 6/20 0.50
GAA P10253 4/20 0.50
MEN1 O00255 3/20 0.50
NPC1 O15118 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1887021 0.87 MAPT (0.67) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL8680075 0.86 KMT2A (0.53) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL5692466 0.83 SMN1; SMN2 (0.57) KMT2AMAPTALDH1A1GAAMEN1
SCHEMBL1184803 0.83 KMT2A (0.50) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL12235984 0.81 MAPT (0.51) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL31150253 0.81 KMT2A (0.51) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL5038742 0.78 ALDH1A1 (0.56) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL29514133 0.78 MAPT (0.51) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL965802 0.78 MAPT (0.51) KMT2AMAPTKDM4EALDH1A1GAA
SCHEMBL30506422 0.77 KMT2A (0.57) KMT2AMAPTKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9018209-B2 Compounds and methods for the treatment of viruses and cancer YALE UNIVERSITY (US) 2015-04-28 US disclosed
US-20110105436-A1 HETEROARYL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE IN CANCER TREATMENT AUCKLAND UNISERVICES LIMITED (NZ) 2011-05-05 US disclosed
US-20100222352-A1 Compounds and Methods for the Treatment of Viruses and Cancer YALE UNIVERSITY (US) 2010-09-02 US disclosed
WO-2009114552-A1 HETEROARYL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE IN CANCER TREATMENT THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2009-09-17 WO disclosed
WO-2007038387-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OF VIRUSES AND CANCER YALE UNIVERSITY (US) 2007-04-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105436-A1 HETEROARYL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE IN CANCER TREATMENT VHL, TP53, BECN1 KMT2A 2132/4885MAPT 2506/4885KDM4E 2441/4885
US-20100222352-A1 Compounds and Methods for the Treatment of Viruses and Cancer RCOR1, RCOR3, CCNT1 KMT2A 2381/4885MAPT 1838/4885KDM4E 3001/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.