SCHEMBL18851069

SCHEMBL18851069

Bc1cc2cc(Cl)ccc2n1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 10/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ROCK2 O75116 1/20 0.38
CHEK2 O96017 1/20 0.38
PRKACA P17612 1/20 0.38
RPS6KA3 P51812 1/20 0.38
PAK1 Q13153 1/20 0.38
ROCK1 Q13464 1/20 0.38
DYRK1A Q13627 1/20 0.38
PRKD2 Q9BZL6 1/20 0.38
NR1H3 Q13133 2/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
GABRA1 P14867 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28106960 0.89 NR1H2 (0.39) NR1H2MEN1KMT2AROCK2CHEK2
SCHEMBL4389624 0.84 AKR1C3 (0.49) NR1H2MEN1KMT2ANR1H3AKR1C3
SCHEMBL13191270 0.83 NR1H2 (0.43) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL17226217 0.82 NR1H2 (0.47) NR1H2AKR1C3AKR1C2ALDH1A1HPGD
SCHEMBL7913537 0.81 NR1H2 (0.56) NR1H2NR1H3CA12CA9
SCHEMBL19013549 0.81 NR1H2 (0.41) NR1H2MEN1KMT2AROCK2CHEK2
SCHEMBL29955454 0.81 NR1H2 (0.39) NR1H2MEN1KMT2AROCK2CHEK2
SCHEMBL29631993 0.81 NR1H2 (0.41) NR1H2MEN1KMT2AROCK2CHEK2
SCHEMBL18990363 0.81 NR1H2 (0.40) NR1H2MEN1KMT2AROCK2CHEK2
SCHEMBL2930214 0.81 NR1H2 (0.39) NR1H2MEN1KMT2AROCK2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017075694-A1 ANTIBIOTIC COMPOUNDS, PHARMACEUTICAL FORMULATIONS THEREOF AND METHODS AND USES THEREFOR SIMON FRASER UNIVERSITY (CA) 2017-05-11 WO disclosed