SCHEMBL28106960

SCHEMBL28106960

Bc1cc2ccc(Cl)cc2n1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 10/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CCR9 P51686 2/20 0.38
NR1H3 Q13133 3/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
STS P08842 1/20 0.36
ROCK2 O75116 1/20 0.36
CHEK2 O96017 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KA3 P51812 1/20 0.36
PAK1 Q13153 1/20 0.36
ROCK1 Q13464 1/20 0.36
DYRK1A Q13627 1/20 0.36
PRKD2 Q9BZL6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18851069 0.89 NR1H2 (0.40) NR1H2MEN1KMT2ANR1H3CA12
SCHEMBL17022491 0.84 NR1H2 (0.40) NR1H2MEN1KMT2ACCR9NR1H3
SCHEMBL13515283 0.84 AKR1C3 (0.40) NR1H2MEN1KMT2ACCR9NR1H3
SCHEMBL17433471 0.83 USP30 (0.44) NR1H2CCR9NR1H3CA12CA9
SCHEMBL24077249 0.82 NR1H2 (0.46) NR1H2CCR9NR1H3ALDH1A1STS
SCHEMBL19013262 0.82 CCR9 (0.51) NR1H2MEN1KMT2ACCR9NR1H3
SCHEMBL7913537 0.81 NR1H2 (0.56) NR1H2NR1H3CA12CA9
SCHEMBL18990058 0.81 NR1H2 (0.40) NR1H2MEN1KMT2ACCR9NR1H3
SCHEMBL18989952 0.81 NR1H2 (0.41) NR1H2MEN1KMT2ACCR9NR1H3
SCHEMBL1605189 0.81 NR1H2 (0.38) NR1H2MEN1KMT2ACCR9NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104193725-B Organic compound 诺华股份有限公司 2016-11-16 CN disclosed