SCHEMBL18856467

SCHEMBL18856467

CS/C(=N\C#N)Nc1ccc(Br)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
MAOB P27338 1/20 0.36
RAB9A P51151 4/20 0.33
MAPT P10636 4/20 0.33
NPC1 O15118 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KIF11 P52732 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18856789 0.84 CYP1A2 (0.48) IDO1RAB9AMAPTNPC1MEN1
SCHEMBL18856804 0.84
SCHEMBL15544661 0.83 KMT2A (0.47) IDO1RAB9AMAPTNPC1MEN1
SCHEMBL15544664 0.83 KMT2A (0.47) IDO1RAB9AMAPTNPC1MEN1
SCHEMBL15606457 0.83 CYP1A2 (0.30) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL19069842 0.83 IDO1 (0.32) IDO1RAB9AKMT2ACYP1A2CYP3A4
SCHEMBL20108715 0.82
SCHEMBL4104086 0.81 ALDH1A1 (0.43) IDO1MAOBRAB9AMAPTNPC1
SCHEMBL4092695 0.81 ALDH1A1 (0.43) IDO1MAOBRAB9AMAPTNPC1
SCHEMBL18856832 0.80 MEN1 (0.30) MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870143-B1 TRIAZOLE COMPOUNDS AS ANTIVIRALS HOFFMANN LA ROCHE (CH) 2017-05-17 EP disclosed