SCHEMBL18890281

SCHEMBL18890281

CC(C)(C)c1cc(-c2cccc(-c3cc(C(C)(C)C)cc(C(C)(C)C)c3O)n2)c(O)c(C(C)(C)C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.56
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
CA2 P00918 3/20 0.42
CA1 P00915 1/20 0.38
GABRA1 P14867 2/20 0.38
GABRB2 P47870 2/20 0.38
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
TYR P14679 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALOX5 P09917 1/20 0.36
PTGS2 P35354 1/20 0.36
PTPN5 P54829 1/20 0.36
GAA P10253 1/20 0.35
XBP1 P17861 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24359601 0.90 HSP90AA1 (0.50) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL17268865 0.83 CA2 (0.55) HSP90AA1CYP1A2CYP2C9TSHRCYP2C19
SCHEMBL1003882 0.83 HSP90AA1 (0.47) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL24359571 0.83 HSP90AA1 (0.44) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL30178546 0.83 HSP90AA1 (0.49) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL14821700 0.83 HSP90AA1 (0.49) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL30646078 0.83 HSP90AA1 (0.41) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL956042 0.81 HSP90AA1 (0.45) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL29671062 0.80 HSP90AA1 (0.62) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR
SCHEMBL29370116 0.80 HSP90AA1 (0.62) HSP90AA1CYP1A2CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170152344-A1 FUNCTIONAL GRAPHENE NANOSTRUCTURE DEVICES FROM LIVING POLYMERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-06-01 US disclosed