SCHEMBL18891798

SCHEMBL18891798

Cc1ccc2cc(C)c(C(C)OC(C)(C)C)c(-c3ccc(Cl)cc3)c2c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.34
CYP3A4 P08684 1/20 0.33
DHODH Q02127 2/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.31
TP53 P04637 2/20 0.30
MAPT P10636 2/20 0.30
CSNK2A2 P19784 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30
PTGS2 P35354 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18892272 0.84 CYP3A4 (0.33) PSIP1CYP3A4
SCHEMBL18892354 0.83 CYP3A4 (0.32) CYP3A4
SCHEMBL1699335 0.83 PSIP1 (0.50) PSIP1CYP3A4DHODHPTGDR2
SCHEMBL15165201 0.83 PSIP1 (0.41) PSIP1CYP3A4DHODHPTGDR2TP53
SCHEMBL18891823 0.82
SCHEMBL18892399 0.80
SCHEMBL18892111 0.79 KCNH2 (0.32) PSIP1PTGDR2TP53ALOX15TSHR
SCHEMBL18892434 0.79
SCHEMBL18892432 0.78
SCHEMBL18892409 0.77 TNIK (0.33) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588450-B1 NAPHT-2-YLACETIC ACID DERIVATIVES TO TREAT AIDS GILEAD SCIENCES INC (US) 2017-05-24 EP disclosed