SCHEMBL18900596

SCHEMBL18900596

CC(C)(C)c1nc(N2CCCC2)c2ccn(Cc3ccccc3S(C)(=O)=O)c2n1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 15/20 0.55
CNR1 P21554 2/20 0.54
HRH3 Q9Y5N1 3/20 0.44
FYN P06241 2/20 0.41
SRC P12931 2/20 0.41
FLT3 P36888 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18557435 0.91 CNR2 (0.53) CNR2CNR1HRH3SRCFLT3
SCHEMBL16212322 0.86 CNR2 (0.74) CNR2CNR1
SCHEMBL16212406 0.86 CNR2 (0.74) CNR2CNR1
SCHEMBL16212404 0.86 CNR2 (0.74) CNR2CNR1
SCHEMBL16212191 0.85 CNR2 (0.64) CNR2CNR1
SCHEMBL18900887 0.82 CNR2 (0.55) CNR2CNR1HRH3FYNSRC
SCHEMBL18900884 0.80 HRH3 (0.47) CNR2CNR1HRH3FYNSRC
SCHEMBL18900883 0.80 CNR2 (0.54) CNR2CNR1HRH3FYNSRC
SCHEMBL18557434 0.76 CNR2 (0.51) CNR2CNR1HRH3SRCFLT3
SCHEMBL18900741 0.75 CNR2 (0.55) CNR2CNR1HRH3FYNSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991988-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CB2 RECEPTOR AGONISTS HOFFMANN LA ROCHE (CH) 2017-05-31 EP disclosed