SCHEMBL18909474

SCHEMBL18909474

CCN1CCC[C@H](C#N)C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.44
DRD2 P14416 2/20 0.44
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NLRP3 Q96P20 2/20 0.34
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
CASP1 P29466 1/20 0.33
L3MBTL3 Q96JM7 1/20 0.33
KDM2B Q8NHM5 1/20 0.33
HTR2A P28223 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15998481 1.00 DRD3 (0.44) DRD3DRD2CYP3A4CYP2D6CYP1A2
SCHEMBL18513114 1.00 DRD3 (0.44) DRD3DRD2CYP3A4CYP2D6CYP1A2
SCHEMBL9870758 0.88
SCHEMBL24661958 0.88
SCHEMBL24662678 0.88
SCHEMBL24789538 0.84 HRH3 (0.39) DRD3DRD2CYP2D6KDM4E
SCHEMBL16625964 0.82 BCHE (0.44) DRD3DRD2CYP2D6TSHRNFKB1
SCHEMBL27282850 0.79 PIK3CD (0.39) KDM4EL3MBTL3
SCHEMBL27281627 0.79 PIK3CD (0.39) KDM4EL3MBTL3
SCHEMBL27284616 0.79 PIK3CD (0.39) KDM4EL3MBTL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017089390-A1 JANUS KINASES INHIBITORS, COMPOSITIONS THEREOF AND USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-01 WO disclosed