SCHEMBL18930700

SCHEMBL18930700

C=CC(C)(C#N)OC(=O)N[C@@H](CCN1CCN(C)CC1)Cc1ccc(C#N)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.36
KCNJ1 P48048 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
SLC1A2 P43004 2/20 0.36
SLC1A3 P43003 1/20 0.36
CCR5 P51681 3/20 0.35
CCR2 P41597 1/20 0.35
HTR1A P08908 5/20 0.35
DRD2 P14416 4/20 0.35
ACACB O00763 1/20 0.34
P2RX7 Q99572 1/20 0.34
HRH1 P35367 4/20 0.34
DRD4 P21917 3/20 0.34
HTR2A P28223 3/20 0.34
OPRM1 P35372 3/20 0.34
HRH2 P25021 3/20 0.34
KCNA5 P22460 2/20 0.34
CACNA1F O60840 2/20 0.34
ADORA3 P0DMS8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18930771 0.88 ATM (0.43) KCNH2KCNJ1ITGB3ITGA2BSLC1A2
SCHEMBL18930522 0.81 ATM (0.43) KCNH2SLC1A2SLC1A3DRD2P2RX7
SCHEMBL18930525 0.80 ACACB (0.45) KCNH2ACACBP2RX7HRH1HRH2
SCHEMBL21144688 0.80 KCNH2 (0.46) KCNH2KCNJ1ITGB3ITGA2BSLC1A2
SCHEMBL21144685 0.80 KCNH2 (0.46) KCNH2KCNJ1ITGB3ITGA2BSLC1A2
SCHEMBL21144891 0.76 ATM (0.40) DRD2P2RX7HRH1HRH2
SCHEMBL21144890 0.76 ATM (0.40) DRD2P2RX7HRH1HRH2
SCHEMBL21169852 0.76 GPR119 (0.42) DRD2P2RX7HRH1HRH2
SCHEMBL18930773 0.76 GPR119 (0.42) DRD2P2RX7HRH1HRH2
SCHEMBL21144689 0.76 ATM (0.40) DRD2P2RX7HRH1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3383865-B1 FURANE DERIVATIVES AS INHIBITORS OF ATAD2 Bayer Pharma AG (DE) 2020-01-29 EP disclosed
WO-2017093272-A1 FURANE DERIVATIVES AS INHIBITORS OF ATAD2 BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-08 WO disclosed