SCHEMBL18939701

SCHEMBL18939701

C=C/C=C(\CC)NCCCNC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 1/20 0.48
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
CA1 P00915 10/20 0.43
CA2 P00918 9/20 0.43
CA12 O43570 7/20 0.43
CA9 Q16790 6/20 0.43
STK17B O94768 1/20 0.39
STK17A Q9UEE5 1/20 0.39
EPHX1 P07099 1/20 0.37
HTT P42858 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19978199 0.80 CA1 (0.35) TDP1MEN1KMT2AGAACA1
SCHEMBL18940165 0.79 TDP1 (0.47) TDP1MEN1KMT2AGAAMAOA
SCHEMBL569251 0.79 TDP1 (0.74) TDP1MEN1KMT2AGAAMAOA
SCHEMBL22169354 0.78 TDP1 (0.35) TDP1MEN1KMT2AGAAMAOA
SCHEMBL18681191 0.77 IDO1 (0.43) TDP1MEN1KMT2AGAAMAOA
SCHEMBL15575825 0.76 TDP1 (0.57) TDP1MEN1KMT2AGAAMAOA
SCHEMBL17934110 0.76 TDP1 (0.61) TDP1MEN1KMT2AGAAMAOA
SCHEMBL18100118 0.75 TDP1 (0.56) TDP1MEN1KMT2AGAAMAOA
SCHEMBL18938501 0.75 TDP1 (0.49) TDP1MEN1KMT2AGAAMAOA
SCHEMBL3020258 0.75 TDP1 (0.81) TDP1MEN1KMT2AGAAMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017096045-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. (US) 2017-06-08 WO disclosed