SCHEMBL18944288

SCHEMBL18944288

CCCCCCCCCNCC1CCC(C(=O)C2CCc3cnn(C)c3Nc3cc(Cl)ccc32)CC1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
GNAI3 P08754 2/20 0.31
GNAO1 P09471 2/20 0.31
GNAI1 P63096 2/20 0.31
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
TSPO P30536 1/20 0.31
MDM2 Q00987 2/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1496096 0.81 IDH1 (0.43) TP53TSPO
SCHEMBL1495933 0.67 AVPR1A (0.42) DRD2TP53
SCHEMBL1496069 0.65 AVPR1A (0.42) DRD3
SCHEMBL2704306 0.64 IDH1 (0.41) TSPO
SCHEMBL2629001 0.62 IDH1 (0.37)
SCHEMBL8597653 0.59 GNAI3 (0.57) DRD2DRD1DRD4DRD5DRD3
SCHEMBL8597657 0.59 GNAI3 (0.57) DRD2DRD1DRD4DRD5DRD3
SCHEMBL19414059 0.58 GNAI3 (0.72) GNAI3GNAO1GNAI1
SCHEMBL11539085 0.58 GNAI3 (0.72) GNAI3GNAO1GNAI1
SCHEMBL1933069 0.58 GNAI3 (0.72) GNAI3GNAO1GNAI1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed