SCHEMBL18944366

SCHEMBL18944366

CN1CCN(c2ccc#cn2)CC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 7/20 0.43
HTR3E A5X5Y0 4/20 0.43
HTR3B O95264 4/20 0.43
HTR3D Q70Z44 4/20 0.43
HTR3C Q8WXA8 4/20 0.43
HRH4 Q9H3N8 6/20 0.41
HRH3 Q9Y5N1 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
THPO P40225 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6068632 0.74 HTR3A (0.51) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL932525 0.70 HRH4 (0.45) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL934301 0.70 HRH4 (0.49) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL1248367 0.70 HTR3A (0.43) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL2068821 0.69 HTR3A (0.46) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL16741177 0.68 HTR3A (0.56) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL1284202 0.66 HRH4 (0.44) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL82036 0.65 HTR3A (0.55) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL16451233 0.65 GAA (0.47) HTR3AKDM4EALDH1A1
SCHEMBL16134879 0.64 CYP1A2 (0.57) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed