SCHEMBL1895899

SCHEMBL1895899

COc1ccc(-n2nc(OCCCN3CCCC3)cc2C)cc1.COc1ccc(-n2nc(OCCN3CCCC3)cc2C)cc1.COc1ccc(-n2nc(OCCN3CCCCC3)cc2C)cc1.COc1ccc(-n2nc(OCCn3ccnc3)cc2C)cc1.Clc1ccc(-n2nc(OCCCN3CCCC3)cc2-c2ccccc2)cc1Cl.Clc1ccc(-n2nc(OCCN3CCCC3)cc2-c2ccccc2)cc1Cl.Clc1ccc(-n2nc(OCCN3CCOCC3)cc2-c2ccccc2)cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.61
KCNH2 Q12809 1/20 0.56
HTR2B P41595 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5182418 0.81 SIGMAR1 (0.94) SIGMAR1KCNH2HTR2B
SCHEMBL5184453 0.79 SIGMAR1 (0.58) SIGMAR1KCNH2
SCHEMBL467012 0.78 SIGMAR1 (1.00) SIGMAR1KCNH2HTR2B
SCHEMBL467378 0.78 SIGMAR1 (0.71) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL1895222 0.78 SIGMAR1 (0.98) SIGMAR1KCNH2HTR2B
Hydrochloric Acid SCHEMBL1897409 0.78 SIGMAR1 (0.70) SIGMAR1KCNH2
SCHEMBL467018 0.77 SIGMAR1 (0.74) SIGMAR1KCNH2
SCHEMBL467024 0.77 SIGMAR1 (0.81) SIGMAR1KCNH2
SCHEMBL467083 0.76 SIGMAR1 (0.83) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL1897470 0.75 SIGMAR1 (0.81) SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2325174-A1 Sigma receptor inhibitors Laboratorios Del. Dr. Esteve, S.A. (ES) 2011-05-25 EP claimed