SCHEMBL18966976

SCHEMBL18966976

Cc1ccc2[nH]c(O)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
KMT2A Q03164 3/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
DAO P14920 2/20 0.44
ALDH1A1 P00352 2/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
PIN1 Q13526 2/20 0.42
GAA P10253 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NQO2 P16083 1/20 0.41
POLB P06746 1/20 0.41
DDO Q99489 1/20 0.41
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947574 0.84 ALDH1A1 (0.61) CYP1A2KMT2AMAPTALDH1A1USP2
SCHEMBL12540 0.79 ALDH1A1 (0.50) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL1171203 0.79 NPC1 (0.51) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL28151599 0.79 PLAU (0.46) KMT2AMAPTMEN1ALDH1A1USP2
Methyl Alcohol SCHEMBL4797570 0.77 CYP1A2 (0.46) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL11268351 0.77 TLR8 (0.39)
SCHEMBL229607 0.76 KMT2A (0.44) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL4441068 0.76 KMT2A (0.51) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL22800202 0.76 KMT2A (0.44) CYP1A2KMT2AMAPTMEN1CYP2C9
SCHEMBL4386728 0.76 KMT2A (0.44) CYP1A2KMT2AMAPTMEN1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017098421-A1 BENZOTHIADIAZINE COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-06-15 WO disclosed