SCHEMBL18970974

SCHEMBL18970974

N[C@@H]1C2CC[C@H]1CN(c1cc(C(F)(F)F)ncn1)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.42
CHKA P35790 1/20 0.42
ACACB O00763 1/20 0.42
PARP1 P09874 1/20 0.38
LCAT P04180 2/20 0.38
DPP4 P27487 5/20 0.35
PSEN1 P49768 7/20 0.35
PSEN2 P49810 7/20 0.35
APH1B Q8WW43 7/20 0.35
NCSTN Q92542 7/20 0.35
APH1A Q96BI3 7/20 0.35
PSENEN Q9NZ42 7/20 0.35
AR P10275 1/20 0.34
KCNH2 Q12809 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
TAF1 P21675 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP7 Q9UHL4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18952546 1.00 CA2 (0.42) CA2CHKAACACBPARP1LCAT
SCHEMBL21726855 1.00 CA2 (0.42) CA2CHKAACACBPARP1LCAT
SCHEMBL21726853 1.00 CA2 (0.42) CA2CHKAACACBPARP1LCAT
SCHEMBL21726804 0.81 DPP4 (0.36) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL18952597 0.81 DPP4 (0.36) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL18952596 0.81 DPP4 (0.36) DPP4PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL2273587 0.79 KDR (0.45) CA2CHKAACACBPARP1LCAT
SCHEMBL20609175 0.78 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL18971472 0.78 PSEN1 (0.39) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL20609161 0.78 PSEN1 (0.39) DPP4PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3386978-B1 BRIDGED PIPERIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2021-01-27 EP disclosed
WO-2017097728-A1 BRIDGED PIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2017-06-15 WO disclosed