SCHEMBL1897341

SCHEMBL1897341

O=C(c1ccc(Cl)c(-c2ccc3cc(O)ccc3c2)c1)N1CCOCC1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.59
HPGD P15428 3/20 0.53
KMT2A Q03164 1/20 0.49
PHGDH O43175 1/20 0.49
KDM4E B2RXH2 1/20 0.48
ABL1 P00519 1/20 0.48
ERN1 O75460 2/20 0.47
CHEK1 O14757 1/20 0.47
PRKCZ Q05513 1/20 0.47
AKR1C3 P42330 1/20 0.45
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
HSP90AA1 P07900 2/20 0.44
HSP90AB1 P08238 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494826 0.84 HPGD (0.59) PKMHPGDKMT2APHGDHHSP90AA1
SCHEMBL18961647 0.81 ERN1 (0.53) PKMHPGDKMT2APHGDHKDM4E
SCHEMBL1901121 0.81 ERN1 (0.76) PKMHPGDKMT2AERN1
SCHEMBL2786906 0.74 HPGD (0.73) PKMHPGDKMT2APHGDHKDM4E
SCHEMBL487574 0.73 PKM (0.77) PKMHPGDKMT2APHGDHKDM4E
SCHEMBL16079573 0.73 KDM4E (0.75) PKMHPGDKMT2APHGDHKDM4E
SCHEMBL12675424 0.73 ERN1 (0.76) PKMHPGDERN1
SCHEMBL2199279 0.72 PHGDH (0.71) PKMHPGDKMT2APHGDHKDM4E
SCHEMBL16592967 0.72 ERN1 (0.60) PKMHPGDPHGDHERN1AKR1C3
SCHEMBL2378698 0.72 PKM (0.75) PKMHPGDKMT2APHGDHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496230-A1 IRE-1 ALPHA INHIBITORS MannKind Corporation (US) 2012-09-12 EP disclosed
WO-2011056744-A1 IRE-1 α INHIBITORS MANNKIND CORPORATION (US) 2011-05-12 WO disclosed