SCHEMBL18976245

SCHEMBL18976245

COC(=O)CCCOc1cc([N+](=O)[O-])c(C(=O)N2CCC[C@H]2C)cc1F

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.42
POLB P06746 1/20 0.42
ALDH1A1 P00352 7/20 0.39
KDM4E B2RXH2 5/20 0.39
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
HRH3 Q9Y5N1 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
GPR174 Q9BXC1 1/20 0.35
THRB P10828 1/20 0.35
KCNK3 O14649 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22272706 0.90 KDM4E (0.43) HPGDPOLBALDH1A1KDM4ECYP2D6
SCHEMBL18976237 0.89 HCRTR1 (0.41) ALDH1A1KDM4ECYP2D6CYP2C19RAB9A
SCHEMBL31717615 0.89 HCRTR1 (0.41) ALDH1A1KDM4ECYP2D6CYP2C19RAB9A
SCHEMBL3931727 0.79 KDM4E (0.41) POLBKDM4ENPC1LMNA
SCHEMBL14072136 0.79 KDM4E (0.41) POLBKDM4ENPC1LMNA
SCHEMBL18953095 0.79 HCRTR1 (0.44) POLBALDH1A1KDM4ECYP2D6CYP2C19
SCHEMBL20581205 0.79 HCRTR1 (0.44) POLBALDH1A1KDM4ECYP2D6CYP2C19
SCHEMBL20975309 0.78 KDM4E (0.43) POLBALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL20975307 0.78 KDM4E (0.43) POLBALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL21000134 0.78 FKBP1A (0.43) POLBKDM4EKMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017098257-A1 PBD ANTIBACTERIAL AGENTS KING'S COLLEGE LONDON (GB) 2017-06-15 WO disclosed